TC-G 1004（化合物 16j）是一种具有口服活性的 A2A 腺苷受体拮抗剂，对 hA2A 和 hA1 的 Ki 值分别为 0.44 nM 和 80 nM。
| Cas No. | 1061747-72-5 |
| 化学名 | N-(2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-(6-(4-methoxypiperidin-1-yl)pyridin-2-yl)pyrimidin-4-yl)acetamide |
| Canonical SMILES | O=C(C)NC1=CC(C2=CC=CC(N3CCC(CC3)OC)=N2)=NC(N4N=C(C)C=C4C)=N1 |
| 分子式 | C22H27N7O2 |
| 分子量 | 421.5 |
| 溶解度 | <42.15mg/ml in 1eq. HCl;<42.15mg/ml in DMSO |
| 储存条件 | Store at -20°C |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request |
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