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Etonogestrel-d6
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Etonogestrel-d6图片
包装与价格:
包装价格(元)
100mg电议
250mg电议
500mg电议

产品名称
3-Oxodesogestrel-d6
3-keto-Desogestrel-d6
产品介绍
Etonogestrel-d6 是 Etonogestrel 氘代物。Etonogestrel (3-Oxodesogestrel) 是孕激素去氧孕烯的生物活性代谢物,Etonogestrel 与靶器官中的孕酮受体 (progesterone receptor) 和雌激素受体 (estrogen receptors) 高亲和力地结合。Etonogestrel 诱导FKBP51mRNA 和蛋白表达
生物活性

Etonogestrel-d6 is deuterium labeled Etonogestrel. Etonogestrel (3-Oxodesogestrel), a biologically active metabolite of progestin Desogestrel, binds with high affinity to progesterone receptors and estrogen receptors in the target organs[1]. Etonogestrel induce FKBP51 mRNA and protein expression in cultured human endometrial stromal cells (HESCs)[2].

体外研究
(In Vitro)

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1].

分子量

330.49

Formula

C22H22D6O2

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.