RKI-1313 是一种ROCK抑制剂，对 ROCK 1 和 ROCK 2 的IC50s 分别为 34、8 μM。RKI-1313 对 ROCK 底物的磷酸化水平、迁移、侵袭或不依赖锚定的生长显示较小的影响。
| 生物活性 | RKI-1313 is aROCKinhibitor withIC50s of 34, 8 μM forROCK1 andROCK2, respectively. RKI-1313 shows little effect on the phosphorylation levels ofROCKsubstrates, migration, invasion or anchorage-independent growth[1]. |
| IC50& Target[1] | ROCK1 34 μM (IC50) | ROCK2 8 μM (IC50) |
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | | Powder | -20°C | 3 years | | In solvent | -80°C | 6 months | | -20°C | 1 month |
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