GW 803430 (GW-3430) 是一种有效的选择性黑色素浓缩激素受体 1 (MCH R1) 拮抗剂,pIC50 为 9.3。
Cas No. | 515141-51-2 |
别名 | GW-3430 |
化学名 | 6-(4-chlorophenyl)-3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)thieno[3,2-d]pyrimidin-4(3H)-one |
Canonical SMILES | ClC1=CC=C(C=C1)C2=CC(N=CN(C3=O)C4=CC=C(C(OC)=C4)OCCN5CCCC5)=C3S2 |
分子式 | C25H24ClN3O3S |
分子量 | 481.99 |
溶解度 | DMF: 2 mg/ml,DMSO: 2 mg/ml,Ethanol: 2 mg/ml,PBS (pH 7.2): Slightly soluble |
储存条件 | Store at -20℃ |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |