CAS NO: | 155584-74-0 |
包装 | 价格(元) |
100mg | 电议 |
250mg | 电议 |
500mg | 电议 |
生物活性 | VUF10166 is a potent and high-affinity5-HT3receptorantagonist, withKivalues of 0.04 nM (5-HT3A) and 22 nM (5-HT3AB). VUF10166 inhibits 5-HT-induced responses at 5-HT3A and 5-HT3AB receptors at nanomolar concentrations. At5-HT3receptor, VUF10166 at higher concentrations also acts as a partial agonist, with anEC50of 5.2 μM[1]. | ||
IC50& Target |
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分子量 | 262.74 | ||
Formula | C13H15ClN4 | ||
CAS 号 | 155584-74-0 | ||
运输条件 | Room temperature in continental US; may vary elsewhere. | ||
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |