CAS NO: | 185376-97-0 |
包装 | 价格(元) |
100mg | 电议 |
250mg | 电议 |
500mg | 电议 |
生物活性 | RS-102221 is a selective5-HT2C receptorantagonist (Ki=10 nM). RS-102221 shows nearly 100-fold selectivity for the5-HT2C receptoras compared to the5-HT2Aand5-HT2B receptors. RS-102221 can promote the differentiation of new nerve cells. RS-102221 increases food-intake and weight-gain in rats[1][2]. | ||||||||
IC50& Target[1] |
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体外研究 (In Vitro) | RS102221 (0.3-300nM; 24 h) 促进小鼠成年海马神经前体细胞 (ahNPCs) 分化,并显著增加 MAP-2+细胞的百分比[1]。 Cell Differentiation Assay[1]
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体内研究 (In Vivo) | RS-102221 (2 mg/kg; 腹腔注射; 每天 1 次, 共 14 天) 增加大鼠的食物摄入量和体重增加[2]。 | ||||||||
分子量 | 612.62 | ||||||||
Formula | C27H31F3N4O7S | ||||||||
CAS 号 | 185376-97-0 | ||||||||
运输条件 | Room temperature in continental US; may vary elsewhere. | ||||||||
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |