5-HT6/5-HT2A receptor ligand-2 (化合物 42) 是一种可透过血脑屏障的5-HT6/5-HT2A的双拮抗剂 ,Ki值分别为 25 nM 和 32 nM。5-HT6/5-HT2A receptor ligand-2 具有促认知特性。
生物活性 | 5-HT6/5-HT2A receptor ligand-2 (compound 42) is a brain-penetrant dual5-HT6/5-HT2Areceptorantagonist, with aKiof 25 nM and 32 nM, respectively. 5-HT6/5-HT2A receptor ligand-2 shows pro-cognitive properties[1]. |
IC50& Target[1] | 5-HT6Receptor 25 nM (Ki) | 5-HT2AReceptor 32 nM (Ki) |
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运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |