CAS NO: | 2244579-87-9 |
包装 | 价格(元) |
5mg | 电议 |
10mg | 电议 |
生物活性 | CB2R PAM is an orally activecannabinoid type-2 receptors (CB2Rs)positive allosteric modulator. CB2R PAM displays antinociceptive activity in vivo in an experimental mouse model of neuropathic pain[1]. | ||||||||
IC50& Target |
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体外研究 (In Vitro) | CB2R PAM (100 nM) significantly enhances the ability of CP55940 and 2-AG, but not of AEA, to stimulate [35S]GTPγS binding to CB2Rs[1]. | ||||||||
体内研究 (In Vivo) | CB2R PAM (1-20 mg/kg; p.o.) displays antinociceptive activity[1].
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分子量 | 435.33 | ||||||||
Formula | C21H24BrFN2O2 | ||||||||
CAS 号 | 2244579-87-9 | ||||||||
运输条件 | Room temperature in continental US; may vary elsewhere. | ||||||||
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |