CAS NO: | 1314230-75-5 |
包装: | 1mg |
市场价: | 2200元 |
生物活性 | CB2receptor agonist 2 is a potent and selective agonist for theCB2(cannabinoid type 2) receptor with aKiof 8.5 nM.CB2receptor agonist 2 has high affinity and selectivity forCB2[1]. | ||||||||
IC50& Target[1] |
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体外研究 (In Vitro) | CB2 receptor agonist 2 (compound 4g) (1 μM; 72 hours) has very low or no cytotoxicity to Hep-G2 cells[1]. Cell Proliferation Assay[1]
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体内研究 (In Vivo) | CB2 receptor agonist 2 (compound 4g) (1 and 3 mg/kg; 1 hour) is very potent (with maximal effect being reached already at the 1 mg/kg dose) and has antihyperalgesic effects, efficacious also on the first phase of the nocifensive response and strongly reduced by AM630 (CB2-selective antagonist/inverse agonist)[1].
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分子量 | 488.62 | ||||||||
Formula | C30H36N2O4 | ||||||||
CAS 号 | 1314230-75-5 | ||||||||
运输条件 | Room temperature in continental US; may vary elsewhere. | ||||||||
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |