JTP-117968 是选择性的糖皮质激素受体调节剂 (非甾类的 SGRM,IC50值为 6.8 nM),具有改善的转录抑制/转激活解离活性。
生物活性 | JTP-117968, a novel selectiveglucocorticoid receptormodulator (a non-steroidal SGRM,IC50of 6.8 nM), exhibits improved transrepression/transactivation dissociation[1]. |
体外研究 (In Vitro) | JTP-117968 has partial TR activity, but exhibits extremely low TA activity[1].
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运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |