GR 127935 hydrochloride 是一种有效且具有口服活性的 5-HT1D 和 5-HT1B 受体拮抗剂，两种异构体的 pKis 均为 8.5。
| Cas No. | 148642-42-6 |
| 化学名 | N-(4-methoxy-3-(4-methylpiperazin-1-yl)phenyl)-2'-methyl-4'-(5-methyl-1,2,4-oxadiazol-3-yl)-[1,1'-biphenyl]-4-carboxamide hydrochloride |
| Canonical SMILES | O=C(C(C=C1)=CC=C1C2=CC=C(C3=NOC(C)=N3)C=C2C)NC4=CC=C(C(N5CCN(C)CC5)=C4)OC.Cl |
| 分子式 | C29H31N5O3.HCl |
| 分子量 | 534.06 |
| 溶解度 | DMSO: 1 mg/ml,DMSO:PBS (pH 7.2) (1:1): 0.25 mg/ml |
| 储存条件 | Desiccate at RT |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request |
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