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CGRP antagonist 1
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
CGRP antagonist 1图片
CAS NO:1123757-49-2
包装与价格:
包装价格(元)
250mg电议
500mg电议

产品介绍
CGRPantagonist1是高效的CGRP受体拮抗剂,Ki和IC50值分别为35和57nM。
Cas No.1123757-49-2
Canonical SMILESO=C(NC1=CC2=C(C[C@@]3(C4=CC=CN=C4NC3=O)C2)C=C1)CN5C(C6(CCOCC6)C7=C5C=CC=C7)=O
分子式C29H26N4O4
分子量494.54
溶解度Soluble in DMSO
储存条件Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
产品描述

CGRP antagonist 1 is a highly potent CGRP receptor antagonist with a Ki and IC50 of 35 and 57 nM, respectively.

CGRP antagonist 1 is compound 20[1].

[1]. Stump CA, et al. The discovery of highly potent CGRP receptor antagonists. Bioorg Med Chem Lett. 2009 Jan 1;19(1):214-7.